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  • Chem Sci Trans., 2014, 3(3),  pp 1043-1046  

    DOI:10.7598/cst2014.849

    Research Article

    Regioselective Synthesis of Some Thio Analogues of Quinolone Antibacterials via Borate Complex of Quinolone Carboxylic Acid Catalyzed by DABCO under Microwave Irradiation

  • SHADI H. RAEIAT1 and AZAR TAHGHIGHI1,2*
  • 1Department of Chemistry, School of Science, Alzahra University, Vanak, Tehran, Iran
    2Malaria and Vector Research Group (MVRG), Biotechnology Research Center (BRC), Pasteur Institute of Iran, Tehran, Iran
  • Abstract

    Regioselective syntheses of some thio analogues were achieved in this paper. Quinolone carboxylic acid were treated with boric acid in acetic anhydride to produce boron complex, which is then reacted with mercapto compounds to afford quinolone derivatives in high yields.

    Keywords

    Quinolone, Boron complex, DABCO, Regioselective synthesis

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